G-protein coupled receptors

Novel GPCR targets for therapeutic research

The G-protein-coupled receptor (GPCR) superfamily comprises an estimated 600–1,000 members and is the largest known class of molecular targets with proven therapeutic value. Our experienced team of GPCR biologists has generated a highly validated and novel family of GPCR cell line products to enable your discovery programs.

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Cell-based GPCR reporter assays

Access GPCR targets with our GeneBLAzer and Tango FRET cell based assays in dividing or division arrested formats.

Cell-based second messenger assays

View our complete portfolio of calcium flux assays for high content and high throughput screening including the Fluo family of fluorescent dyes.  These indicators provide a rapid method of imaging calcium flux associated with GPCR activation or inhibition.

GPCR antibodies & immunoassays

Find the right GPCR antibody for your research needs.

Membrane protein expression system

Produce functional GPCRs in mammalian cells as virus-like particles (VLPs) for use in receptor-ligand binding or antibody binding studies.

For Research Use Only. Not for use in diagnostic procedures.